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Products > Epigenetics > DNA methyltransferase > LGK-974 (LGK974, LGK 974)
LGK-974 (LGK974, LGK 974)
Product name : LGK-974 (LGK974, LGK 974)
Product No. : cs-1102
Price : 100mg, $675, 500mg/$1875
CAS : 
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  Details:
LGK-974 (CAS: 1243244-14-5) is a potent and specific PORCN inhibitor, and inhibits Wnt signaling with IC50 of 0.4 nM. Porcupine, a membrane-bound O-acyltransferase (MBOAT), is required for the palmitoylation of Wnt ligands, and plays a key role in Wnt ligand secretion and activity. Wnt signaling is dysregulated in a variety of cancers.

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