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Products > PI3K/Akt/mTOR > PI3K > TGR-1202 (RP5264; TGR1202; TGR 1202; RP-5264; RP 5264)
TGR-1202 (RP5264; TGR1202; TGR 1202; RP-5264; RP 5264)
Product name : TGR-1202 (RP5264; TGR1202; TGR 1202; RP-5264; RP 5264)
Product No. : cs-2443
Price : 100mg, $675, 500mg/$1875
CAS : 
Bulk inquiry : 
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  Details:
TGR-1202 (CAS: 1532533-67-7 (free base), 1532533-78-0 (HCL)) is a novel PI3Kδ inhibitor, with IC50 and EC50 of 22.2 nM and 24.3 nM, respectively; Also active against CK1ε, with an EC50 value of 6.0 μM. Inhibition of PI3K delta signaling with TGR-1202 has demonstrated robust activity in numerous pre-clinical models and primary cells from patients with hematologic malignancies.

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