GSK6853 (CAS: 1910124-24-1) is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrated properties suitable for cellular and in vivo studies. The BRPF (Bromodomain and PHD Fingercontaining) protein family are important scaffolding proteins for assembly of MYST histone acetyltransferase complexes.
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Technical Data
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Appearance:
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Off White Solid
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Purity:
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> 98%
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QC Data:
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 View Current Lot Data File
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CAS:
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1910124-24-1
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Storage
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-20°C, long term; 4°C, short term
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Shipping
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Room temperature
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TGF-beta/Smad
Histone Methyltransferase
