TGF-beta/Smad
Aurora Kinase
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Product name : EPZ-011989 (EPZ011989)
Product No. : cs-2079
Price : 100mg, $475, 500mg/$1275
CAS :
Bulk inquiry :
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| Details: |
EPZ011989 (CAS:1598383-40-4) is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. Inhibitors of the protein methyltransferase Enhancer of Zeste Homolog 2 (EZH2) may have significant therapeutic potential for the treatment of B cell lymphomas and other cancer indications.
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