Product name : Enzastaurin (LY317615, LY-317615)
Product No. : cs-1980
Price : 50mg, $675; 100mg, $1175
CAS :
Bulk inquiry :
|
Details: |
LY 317615 (CAS: 170364-57-5) is a potent PKCβ selective inhibitor with IC50 of 6 nM, 6- to 20-fold selectivity against PKCα, PKCγ and PKCε. Binding to the ATP-binding site, enzastaurin selectively inhibits protein kinase C beta, an enzyme involved in the induction of vascular endothelial growth factor (VEGF)-stimulated neo-angiogenesis. This agent may decrease tumor blood supply and so tumor burden.
|
Related Products : |
|
|
|
|
||||||||
|
|
|
|