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Products > Others > Others > GSK-2879552 (GSK2879552, GSK 2879552)
GSK-2879552 (GSK2879552, GSK 2879552)
Product name : GSK-2879552 (GSK2879552, GSK 2879552)
Product No. : cs-1621
Price : 100mg, $675, 500mg/$1875
CAS : 
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  Details:
 GSK2879552 (CAS: 1401966-69-5) is an orally available, irreversible, inhibitor of lysine specific demethylase 1 (LSD1), with potential antineoplastic activity. Upon administration, GSK2879552 binds to and inhibits LSD1, a demethylase that suppresses the expression of target genes by converting the dimethylated form of lysine at position 4 of histone H3 (H3K4) to mono- and unmethylated H3K4. LSD1 inhibition enhances H3K4 methylation and increases the expression of tumor-suppressor genes. This may lead to an inhibition of cell growth in LSD1-overexpressing tumor cells. LSD1, overexpressed in certain tumor cells, plays a key role in tumor cell growth and survival.

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