cckinase, Inc.

Favorite  |  Set Home
E-mail: info@cckinase.com
Products > Metabolic enzyme/Protease > Isocitrate Dehydrogenases > Enasidenib (AG221, AG-221, AG 221)
Enasidenib (AG221, AG-221, AG 221)
Product name : Enasidenib (AG221, AG-221, AG 221)
Product No. : cs-1590
Price : 100mg, $675, 500mg/$1875
CAS : 
Bulk inquiry : 
←[Previous Product]              [Next Product]→
Online Inquiry         Email Us

  Details:
 Enasidenib (CAS: 1446502-11-9) is a oral potent, selective, reversible inhibitor of mutant IDH2. The mutations of IDH2 present in certain cancer cells result in a new ability of the enzyme to catalyze the NAPH-dependent reduction of α-ketoglutarate to R(-)-2-hydroxyglutarate (2HG). The production of 2HG is believed to contribute to the formation and progression of cancer . The inhibition of mutant IDH2 and its neoactivity is therefore a potential therapeutic treatment for cancer. 

  Related Products :

Mutant IDH1-IN-1
Mutant IDH1-IN-1
Price: 50mg, $675; 100mg, $1175

AGI-6780 (AGI6780, AGI 6780)
AGI-6780 (AGI6780, AGI 6780)
Price: 100mg, $475, 500mg/$1275

AGI-6780 (AGI6780)
AGI-6780 (AGI6780)
Price: 100mg, $475, 500mg/$1275

Ivosidenib (AG-120; AG 120; AG120)
Ivosidenib (AG-120; AG 120; AG120)
Price: 100mg, $675, 500mg/$1875

Vorasidenib (AG-881, AG881, AG 881)
Vorasidenib (AG-881, AG881, AG 881)
Price: 50mg/$675, 100mg/$975

Ivosidenib (AG-120, AG120, AG 120)
Ivosidenib (AG-120, AG120, AG 120)
Price: 100mg, $475, 500mg/$1275

LTURM34 (LTURM-34, LTURM 34)
LTURM34 (LTURM-34, LTURM 34)
Price: 50mg/$675, 100mg/$975

DS-1001B
DS-1001B
Price: 100mg/$675; 500mg/$1875

Online service

info@cckinase.com