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Products > Protein Tyrosine Kinase/RTK > BTK > CNX-774 (CNX774; CNX 774)
CNX-774 (CNX774; CNX 774)
Product name : CNX-774 (CNX774; CNX 774)
Product No. : cs-946
Price : 100mg, $675, 500mg/$1875
CAS : 
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  Details:
CNX-774 (CAS: 1202759-32-7) is a potent, selective, and orally available small molecule inhibitor of Btk (IC50< 1 nM) that forms a ligand-directed covalent bond with Cys-481, a non-conserved amino acid within the active site of the enzyme. Bruton's tyrosine kinase (BTK) , a crucial terminal kinase enzyme in the B-cell antigen receptor (BCR) signaling pathway, has emerged as an attractive target for therapeutic intervention in human malignancies and autoimmune disorders.

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